DDR inhibitor X( —— )

Catalog No. M12505 CAS No. 1644069-80-6

COA

Datasheet

HNMR

HPLC

MSDS

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Product Name

DDR inhibitor X
Note

Research use only, not for human use.
Brief Description

DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2.
Description

DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
In Vitro

DDR Inhibitor (Example 6) is a potent DDR inhibitor, with an IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
In Vivo

——
Synonyms

——
Pathway

Tyrosine Kinase
Target

DDR
Recptor

DDR
Research Area

Cancer
Indication

——

CAS Number

1644069-80-6
Formula Weight

417.444
Molecular Formula

C23H20FN5O2
Purity

>98% (HPLC)
Solubility

DMSO : 65 mg/mL 155.71 mM; H2O : < 0.1 mg/mL
SMILES

CC1=C(C=C(C=C1)CNC(=O)NC2=CC(=CC=C2)F)NC(=O)C3=CN=C4N3C=CC=C4
Chemical Name

N-[5-[[[(3-Fluorophenyl)carbamoyl]amino]methyl]-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide

1. Patent WO2015004481A1.

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